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Methylnaltrexone: Benefits, Reviews, Info, Side Effects!
Rx Details
Methylnaltrexone
Relistor, Relistor Subcutaneous, Relistor Oral
Methylnaltrexone
Prescription
Medication
Drugs
Prescription Only
relieves opioid-induced constipation, does not affect pain relief from opioids, works quickly, administered subcutaneously, minimal central nervous system effects
Abdominal Pain, Diarrhea, Dizziness, Flatulence, Gastrointestinal Perforation, Hyperhidrosis, Nausea
Methylnaltrexone is a medication used to treat opioid-induced constipation. The dosage of methylnaltrexone can vary based on the form of the medication and the patient’s specific needs, including their weight and the severity of their condition. For the subcutaneous injection form, the typical dosage is often calculated based on body weight. A common dosage is 0.15 mg per kilogram of body weight, administered every other day as needed, but not more frequently than once every 24 hours. It’s important to note that the exact dosage should be determined by a healthcare professional, who will consider the patient’s overall health, kidney function, and other medications they may be taking. Always follow the prescribing doctor’s instructions or the guidelines provided with the medication.
Opioid-induced constipation
Generally well-tolerated with minimal side effects.
No Interactions Reported
$100 – $200
$1,200

A Synopsis of

Methylnaltrexone

Methylnaltrexone is a medication that is used to treat opioid-induced constipation in patients who are receiving opioid therapy for chronic pain. Opioid medications are commonly prescribed for pain management, but they can also cause constipation as a side effect. Methylnaltrexone works by blocking the effects of opioids in the gut, which helps to alleviate constipation without affecting the pain-relieving effects of the opioids.

This medication is typically administered by injection under the skin, and it works quickly to provide relief from constipation. It is important to follow the dosing instructions provided by your healthcare provider to ensure that you are receiving the appropriate amount of medication for your individual needs.

As with any medication, there are potential side effects associated with methylnaltrexone. These may include abdominal pain, nausea, diarrhea, and dizziness. It is important to discuss any concerns or questions you may have with your healthcare provider before starting this medication.

Overall, methylnaltrexone can be a valuable tool in managing opioid-induced constipation for patients who are on long-term opioid therapy. By addressing this common side effect, patients can experience improved quality of life and better overall health outcomes. If you are experiencing constipation as a result of opioid therapy, talk to your healthcare provider about whether methylnaltrexone may be a suitable treatment option for you.

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The information provided on RxDB.net is for informational purposes only and is not intended to replace professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare professional, such as a doctor or pharmacist, for any questions or concerns regarding your health, medications, or medical conditions. Reliance on any information provided on this website is solely at your own risk. RxDB.net does not provide medical or pharmaceutical services and is not liable for any decisions made based on the information contained herein.

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